Cart
sales@molnova.com
Home - Products - Endocrinology/Hormones - 5-HT Receptor - SB 206553

SB 206553

CAS No. 1197334-04-5

SB 206553 ( SB206553 )

Catalog No. M10703 CAS No. 1197334-04-5

SB 206553 is a potent and selective 5-HT2B/5-HT2C receptor antagonist with pA2 of 8.89 for rat 5-HT2B, pKi of 7.92 for human 5-HT2C, displays >80-fold selectivity over other 5-HT receptor subtypes.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 963 Get Quote
50MG 1962 Get Quote
100MG 2520 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote
Group Booking Get Quotation Bulk Inquiry Add to Cart

Biological Information

  • Product Name
    SB 206553
  • Note
    Research use only, not for human use.
  • Brief Description
    SB 206553 is a potent and selective 5-HT2B/5-HT2C receptor antagonist with pA2 of 8.89 for rat 5-HT2B, pKi of 7.92 for human 5-HT2C, displays >80-fold selectivity over other 5-HT receptor subtypes.
  • Description
    SB 206553 is a potent and selective 5-HT2B/5-HT2C receptor antagonist with pA2 of 8.89 for rat 5-HT2B, pKi of 7.92 for human 5-HT2C, displays >80-fold selectivity over other 5-HT receptor subtypes; exhibits anxiolytic-like properties both in vitro and in vivo.Anxiety Discontinued
  • Synonyms
    SB206553
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    5-HT Receptor
  • Research Area
    Neurological Disease
  • Indication
    Anxiety

Chemical Information

  • CAS Number
    1197334-04-5
  • Formula Weight
    328.80
  • Molecular Formula
    C17H16N4O.HCl
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    O=C(N1C(C(CC1)=C2)=CC3=C2N(C)C=C3)NC4=CC=CN=C4.[H]Cl
  • Chemical Name
    3,5-Dihydro-5-methyl-N-3-pyridinylbenzo[1,2-b:4,5-b']dipyrrole-1(2H)-carboxamide hydrochloride

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Forbes IT, et al. J Med Chem. 1995 Jul 7;38(14):2524-30.
2. Upton N, et al. Eur J Pharmacol. 1998 Oct 16;359(1):33-40.
3. Kennett GA, et al. Br J Pharmacol. 1996 Feb;117(3):427-434.
4. Porras G, et al. Neuropsychopharmacology. 2002 Mar;26(3):311-24.
Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog
related products

  • WAY-100635

    A potent and selective 5-HT1A receptor antagonist; also acts as potent full agonist at the D4 receptor.

  • Fluoxetine hydrochlo...

    Fluoxetine HCl is an antidepressant of the selective serotonin reuptake inhibitor (SSRI) class.

  • SUVN-502 mesylate

    SUVN-502 (SUVN502)is a potent, selective, brain penetrant and orally active 5-HT6 receptor antagonist with Ki of 2.04 nM.

Sign In Join Free